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カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
TP1445 | [Des-Arg9]-Bradykinin acetate | Bradykinin Receptor | |
TP1918L1 | Lys-[Des-Arg9]Bradykinin acetate | Lys-[Des-Arg9]Bradykinin acetate (71800-36-7 free base) | Bradykinin Receptor |
Lys-[Des-Arg9]Bradykinin acetate is an endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and > 30000 nM at human B1 and B2 receptors respectively). Hypotensive agent that reduces p... | |||
TP1917L1 | Sar-[D-Phe8]-des-Arg9-Bradykinin acetate | Sar-[D-Phe8]-des-Arg9-Bradykinin acetate(126959-88-4 free base) | Bradykinin Receptor |
Sar-[D-Phe8]-des-Arg9-Bradykinin acetate is a potent and selective bradykinin B1 receptor agonist (EC50 = 9.02 nM in rabbit aorta) that is resistant to aminopeptidase, kininase I and II (ACE) and neutral endopeptidase cl... | |||
T80072 | Des-Arg9-[Leu8]-Bradykinin acetate | Bradykinin Receptor | |
Des-Arg9-[Leu8]-Bradykinin acetate is a potent antagonist of the bradykinin receptor 1 (B1R), utilized in renal fibrosis research [1]. |